Article citationsMore>>
N. D. Obushak, N. T. Pokhodylo, I. T. Krupa and V. S. Matiichuk, “Synthesis of substituted 4-([1,2,4]triazolo- [3,4-b]-[1,3,4]thiadiazol-6-yl)quinolines,” Russian Journal of Organic Chemistry, Vol. 43, No. 8, 2007, pp. 1223-1227. doi:10.1134/S1070428007080246
has been cited by the following article:
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TITLE:
Highly Efficient Synthesis of Novel Fluorine Bearing Quinoline-4-carboxylic Acid and the Related Compounds as Amylolytic Agents
AUTHORS:
Mohammed S. T. Makki, Dina A. Bakhotmah, Reda M. Abdel-Rahman
KEYWORDS:
Amylolytic Activity; Amylolytic Agents; Aspergillus fungi; Efficient Synthesis; Fluoroquinoline;Quinoline-4-carboxylic Acids
JOURNAL NAME:
International Journal of Organic Chemistry,
Vol.2 No.1,
March
15,
2012
ABSTRACT: Highly efficient syntheses of novel fluorine bearing quinoline-4-carboxylic acids and the related compounds had been achieved from cyclocondensation of 2-amino-5-fluorophenyl glyoxylic acid 1 with benzoyle asetanilides 2 in boiling DMF, to give the target 3. Decarboxylation of 3 produced 6-fluoro-2-phenyl-3-(substituted amino)-keto-quinolines 4, while that reaction underwent refluxing, afforded 7-fluoro-1-(aryl)-3-phenyl-pyrrolo[3,4-c] quinoline-2,9-diones 5. Structure of the products has been established from their elemental and spectral analysis. All targets exhibited a high to moderate activity against some Aspergillus fungi as amylolytic agents.