Article citationsMore>>
Mossine, A.V., Brooks, A.F., Makaravage, K.J., Miller, J.M., Ichlishi, N., Sanford, M.S. and Scott, P.J.H. (2015) Synthesis of [18F]Arenes via the Copper-Mediated [18F]Fluorination of Boronic Acids. Organic Letters, 17, 5780-5783.
https://doi.org/10.1021/acs.orglett.5b02875
has been cited by the following article:
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TITLE:
Effect of Added Cu(OTf)2 on the Cu(OTf)2(Py)4-Mediated Radiofluorination of Benzoyl and Phthaloylglycinates
AUTHORS:
David W. Blevins, George W. Kabalka, Dustin R. Osborne, Murthy R. Akula
KEYWORDS:
Glycinates, Boronate Esters, Gorlos-Phos, Radiofluorination, Copper Triflate
JOURNAL NAME:
Natural Science,
Vol.10 No.3,
March
30,
2018
ABSTRACT: Cu(OTf)2(Py)4 mediated radiofluorination of the boronate esters of
ethyl benzoyl and phthaloylglycinates (11 and 16) using 10 mol% of the copper
complex following the literature procedure did not provide the fluorinated
products. However, the addition of Cu(OTf)2resulted in the radio-fluorination of the boronate esters 11
and 16 to obtain ethyl 4-[18F]fluorobenzoyl glycinate, 17, (48%) and ethyl 3-[18F]phthaloylglycinate (41%) respectively.