Article citationsMore>>
Teare, H., Robins, E.G., Kirjavainen, A., Fordback, S., Sanford, G., Solin, O., Luthra, S.K. and Gouverneur, V. (2010) Radiosynthesis and Evaluation of [18F]Selectfluor Bis(Triflate). Angewandte Chemie International Edition, 122, 6973-6976.
https://doi.org/10.1002/ange.201002310
has been cited by the following article:
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TITLE:
Effect of Added Cu(OTf)2 on the Cu(OTf)2(Py)4-Mediated Radiofluorination of Benzoyl and Phthaloylglycinates
AUTHORS:
David W. Blevins, George W. Kabalka, Dustin R. Osborne, Murthy R. Akula
KEYWORDS:
Glycinates, Boronate Esters, Gorlos-Phos, Radiofluorination, Copper Triflate
JOURNAL NAME:
Natural Science,
Vol.10 No.3,
March
30,
2018
ABSTRACT: Cu(OTf)2(Py)4 mediated radiofluorination of the boronate esters of
ethyl benzoyl and phthaloylglycinates (11 and 16) using 10 mol% of the copper
complex following the literature procedure did not provide the fluorinated
products. However, the addition of Cu(OTf)2resulted in the radio-fluorination of the boronate esters 11
and 16 to obtain ethyl 4-[18F]fluorobenzoyl glycinate, 17, (48%) and ethyl 3-[18F]phthaloylglycinate (41%) respectively.