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Ohtake, Y., Sato, T., Kobayashi, T., Nishimoto, M., Taka, N. and Takano, K. (2012) Discovery of Tofogliflozin, a Novel C-Arylglucoside with an O-Spiroketal Ring System, as a Highly Selective Sodium Glucose Cotransporter 2 (SGLT2) Inhibitor for the Treatment of Type 2 Diabetes. Journal of Medicinal Chemistry, 55, 7828-7840.
https://doi.org/10.1021/jm300884k
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