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Palani, A., Shapiro, S., Josien, H., Bara, T., Clader, J.W., Greenlee, W.J., et al. (2002) Synthesis, SAR, and Biological Evaluation of Oximino-Piperidino-Piperidine Amides. 1. Orally Bioavailable CCR5 Receptor Antagonists with Potent Anti-HIV Activity. Journal of Medicinal Chemistry, 45, 3143-3160.
https://doi.org/10.1021/jm0200815
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